Brian de Costa: шукати на сайті Z-Library

De Costa, Brian R., George, Clifford, Burke, Terrence R., Rafferty, Michael F., Contreras, Patricia C., Mick, Stephen J., Jacobson, Arthur E., Rice, Kenner C.

Рік:

1993

Мова:

english

Файл:

PDF, 865 KB

english, 1993

Synthesis, configuration, and evaluation of two conformationally restrained analogs of phencyclidine

Журнал:

Yoshida, Takeshi, Torsani, Vinicius, Gomes, Susimeire, De Santis, Roberta R., Beraldo, Marcelo A., Costa, Eduardo L. V., Tucci, Mauro R., Zin, Walter A., Kavanagh, Brian P., Amato, Marcelo B. P.

Рік:

1988

Мова:

english

Файл:

PDF, 724 KB

english, 1988

Spontaneous Effort Causes Occult Pendelluft during Mechanical Ventilation

Журнал:

American Journal of Respiratory and Critical Care Medicine

Рік:

2013

Мова:

english

Файл:

PDF, 1.62 MB

english, 2013

Remarkable fly (Diptera) diversity in a patch of Costa Rican cloud forest: Why inventory is a vital science

BORKENT, ART, BROWN, BRIAN V., ADLER, PETER H., AMORIM, DALTON DE SOUZA, BARBER, KEVIN, BICKEL, DANIEL, BOUCHER, STEPHANIE, BROOKS, SCOTT E., BURGER, JOHN, BURINGTON, Z.L., CAPELLARI, RENATO S., COSTA

Журнал:

Zootaxa

Рік:

2018

Мова:

english

Файл:

PDF, 3.19 MB

english, 2018

ChemInform Abstract: Synthesis and Transporter Binding Properties of Bridged Piperazine Analogues of 1-{2-[Bis(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine (GBR 12909).

Ying Zhang, Richard B. Rothman, Christina M. Dersch, Brian R. de Costa, Arthur E. Jacobson, Kenner C. Rice

Журнал:

ChemInform

Рік:

2001

Файл:

PDF, 36 KB

2001

Synthesis of carbon-14 labeled (±)-2-methyl-3,3-diphenyl-3-propanolamine (2-MDP)

Brian De Costa, Andrew Thurkauf, Arthur E. Jacobson, Kenner C. Rice

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1988

Мова:

english

Файл:

PDF, 150 KB

english, 1988

Synthesis of tritium labelled 4-fluoro-1-[1–(2-thienyl)]cyclohexylpiperidine ([3H]-FTCP); a tool for autoradiographic study of the phencyclidine binding site

Andrew Thurkauf, Brian R. De Costa, Dale O. Kiesewetter, Arthur E. Jacobson, Kenner C. Rice

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1989

Мова:

english

Файл:

PDF, 270 KB

english, 1989

Synthesis of high specific activity tritium labelled 1S,2S-(-)-trans-2-isothiocyanato-N-methyl-N-[2-(1-pyrrolidinyl)-cyclohexyl]benzeneacetamide, a specific irreversible ligand for kappa opioid receptors

Brian R. De Costa, Andew Thurkauf, Richard R. Rothman, Arthur E. Jacobson, Kenner C. Rice

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1990

Мова:

english

Файл:

PDF, 383 KB

english, 1990

Synthesis and evaluation of [3H]-4-fluoro-1-[1-(3-hydroxyphenyl)cyclohexyl]piperidine, a potential tool for autoradiographic study of the phencyclidine receptor

Brian R. de Costa, Mariena V. Mattson

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1991

Мова:

english

Файл:

PDF, 554 KB

english, 1991

Synthesis of high specific activity (3,4-[3H]cyclohexyl)-N-[1 (2-benzo[b]thienyl)cyclohexyl]piperidine {[3H]BTCP}: A selective probe for the dopamine-reuptake complex

Brian R. de Costa

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1991

Мова:

english

Файл:

PDF, 455 KB

english, 1991

Synthesis and characterization of optically pure [3H](+)azidophenazocine ([3H](+)-AZPH), a novel photoaffinity label for sigma receptors

Brian R. de Costa, Wayne D. Bowen

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1991

Мова:

english

Файл:

PDF, 551 KB

english, 1991

An expedient synthesis of high specific activity tritium labelled 4-fluoro-1-[1-(2-thienyl)]cyclohexylpiperidine ([3H]FTCP), a ligand for further characterization of the phencyclidine/NMDA receptor complex

Neile A. Grayson, Brian R. de Costa, Joannes T. M. Linders, Kenner C. Rice

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1991

Мова:

english

Файл:

PDF, 319 KB

english, 1991

Synthesis of unlabelled and tritium labelled 4-isothiocyanato-1-(1-phenylcyclohexyl)piperidine (fourphit), tools for the study of the dopamine reuptake complex.

Joannes T. M. Linders, Brian R. de Costa, Neile A. Grayson, Kenner C. Rice

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1992

Мова:

english

Файл:

PDF, 656 KB

english, 1992

Synthesis of [3H]tert-butyl 8-chloro-5,6-dihydro-5-methyl-6-oxo-4h-imidazo[1,5-a][1,4]benzodiazepine 3-carboxylate, a selective, high affinity ligand for the diazepam insensitive (DI) subtype of the benzodiazepine receptor

Zi-Qiang Gu, Brian R. de Costa, Garry Wong, Kenner C. Rice, Phil Skolnick

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1992

Мова:

english

Файл:

PDF, 388 KB

english, 1992

Synthesis of a novel 123I-labelled derivative of GBR12783, a potential agent for SPECT imaging of dopamine-reuptake sites

Xiao-Shu He, Kan Sam Lee, Daniel Weinberger, Brian R. de Costa

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1993

Мова:

english

Файл:

PDF, 408 KB

english, 1993

Synthesis of N1-3-[18F]fluoropropyl-N4-2-([3,4-dichlorophenyl]ethyl)piperazine, a high affinity ligand for sigma receptor

Dale O. Kiesewetter, Brian de Costa

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1993

Мова:

english

Файл:

PDF, 275 KB

english, 1993

A comparison of the incorporation of 123I and 18F into 1-[1-(3-hydroxyphenyl) cyclohexyl]-4-(methanesulfonyloxy)piperidine by nucleophilic displacement with 123I− and 18F−

Xiao-Shu He, Dale O. Kiesewetter, Kan Sam Lee, Mariena V. Mattson, D. R. Weinberger, Brian R. de Costa

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1993

Мова:

english

Файл:

PDF, 474 KB

english, 1993

Synthesis of [123I]tert-butyl 8-iodo-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine 3-carboxylate, a potential SPECT imaging agent for diazepam-insensitive (DI) benzodiazepine receptors

Xiao-Shu He, Dorota Matecka, Kan Sam Lee, Zi-Qiang Gu, Kenner C. Rice, Garry Wong, Phil Skolnick, Brian R. De Costa

Журнал:

Journal of Labelled Compounds and Radiopharmaceuticals

Рік:

1994

Мова:

english

Файл:

PDF, 355 KB

english, 1994

The large-scale polarization of the microwave foreground

Angélica de Oliveira-Costa, Max Tegmark, Christopher O’Dell, Brian Keating, Peter Timbie, George Efstathiou, George Smoot

Журнал:

New Astronomy Reviews

Рік:

2003

Мова:

english

Файл:

PDF, 166 KB

english, 2003

Identification of a GBR12935 homolog, LR1111, which is over 4,000-fold selective for the dopamine transporter, relative to serotonin and norepinephrine transporters

Richard B. Rothman, Bruce Lewis, Chris Dersch, Heng Xu, Lillian Radesca, Brian R. De Costa, Kenner C. Rice, Robert B. Kilburn, Hyacinth C. Akunne, Agu Pert

Журнал:

Synapse

Рік:

1993

Мова:

english

Файл:

PDF, 527 KB

english, 1993

Differential effects of systemically administered nor-binaltorphimine (nor-BNI) on κ-opioid agonists in the mouse writhing assay

Jillian H. Broadbear, S. Stevens Negus, Eduardo R. Butelman, Brian R. de Costa, James H. Woods

Журнал:

Psychopharmacology

Рік:

1994

Мова:

english

Файл:

PDF, 1.22 MB

english, 1994

Microinjection of sigma ligands into cranial nerve nuclei produces vacuous chewing in rats

Thuytien T. Tran, Brian R. de Costa, R. R. Matsumoto

Журнал:

Psychopharmacology

Рік:

1998

Мова:

english

Файл:

PDF, 730 KB

english, 1998

Synthesis and anticonvulsant activity of 1-phenylcyclohexylamine analogs

Thurkauf, Andrew, De Costa, Brian, Yamaguchi, Shunichi, Mattson, Mariena V., Jacobson, Arthur E., Rice, Kenner C., Rogawski, Michael A.

Журнал:

Рік:

1990

Мова:

english

Файл:

PDF, 817 KB

english, 1990

Synthesis and biological evaluation of conformationally restricted 2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylenediamines as .sigma. receptor ligands. 1. Pyrrolidine, piperidine, homopiperidine, and tetrahydroisoquinoline classes

De Costa, Brian R., Dominguez, Celia, He, Xiao Shu, Williams, Wanda, Radesca, Lilian, Bowen, Wayne

Журнал:

He, Xiaoshu, Raymon, Lionel P., Mattson, Mariena V., Eldefrawi, Mohyee E., de Costa, Brian R.

Рік:

1992

Мова:

english

Файл:

PDF, 1.28 MB

english, 1992

Further studies of the structure-activity relationships of 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine. Synthesis and evaluation of 1-(2-benzo[b]thienyl)-N,N-dialkylcyclohexylamines at dopamine uptake and phencyclidine binding sites

Журнал:

Рік:

1993

Мова:

english

Файл:

PDF, 848 KB

english, 1993

Drug specificity of pharmacological dystonia

Rae R. Matsumoto, Mitzi K. Hemstreet, Naline L. Lai, Andrew Thurkauf, Brian R. De Costa, Kenner C. Rice, Susan B. Hellewell, Wayne D. Bowen, J. Michael Walker

Журнал:

Рік:

1990

Мова:

english

Файл:

PDF, 544 KB

english, 1990

GBR12909 antagonizes the ability of cocaine to elevate extracellular levels of dopamine

Richard B. Rothman, Andrea Mele, Audrey A. Reid, Hyacinth C. Akunne, Nigel Greig, Andrew Thurkauf, Brian R. de Costa, Kenner C. Rice, Agu Pert

Журнал:

Рік:

1991

Мова:

english

Файл:

PDF, 1.21 MB

english, 1991

Cocaine and GBR12909 produce equivalent motoric responses at different occupancy of the dopamine transporter

Richard B. Rothman, Nigel Grieg, Andrew Kim, Brian R. de Costa, Kenner C. Rice, F.Ivy Carroll, Agu Pert

Журнал:

William P. Smotherman, Scott R. Robinson, Elena I. Varlinskaya, Evgeniy S. Petrov, Marion Orlowski, Brian R. de Costa, Kenner C. Rice

Рік:

1992

Мова:

english

Файл:

PDF, 801 KB

english, 1992

Central administration of the endopeptidase 24.15 inhibitor cFP-AAF-pAB suggests dynorphin as the endogenous ligand underlying behavioral effects of milk in the fetal rat

Журнал:

European Journal of Pharmacology: Molecular Pharmacology

Рік:

1994

Мова:

english

Файл:

PDF, 505 KB

english, 1994

Site-specific acylation of GABA-gated Cl− channels: effects on 36Cl− uptake

Eric J. Moody, Anita H. Lewin, Brian R. de Costa, Kenner C. Rice, Phil Skolnick

Журнал:

Рік:

1991

Мова:

english

Файл:

PDF, 452 KB

english, 1991

Evidence for mutually exclusive binding of cocaine, BTCP, GBR 12935, and dopamine to the dopamine transporter

Maarten E.A. Reith, Brian de Costa, Kenner C. Rice, Arthur E. Jacobson

Журнал:

European Journal of Pharmacology: Molecular Pharmacology

Рік:

1992

Мова:

english

Файл:

PDF, 778 KB

english, 1992

Differential effects of cytochrome P-450 induction on ligand binding to σ receptors

Anthony S. Basile, Ian A. Paul, Brian de Costa

Журнал:

European Journal of Pharmacology: Molecular Pharmacology

Рік:

1992

Мова:

english

Файл:

PDF, 327 KB

english, 1992

Labelling of diazepam-sensitive and -insensitive benzodiazepine receptors with [3H]tert-butyl-8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazol[1,5-a][1,4]benzodiazepine 3-carboxylate (ZG-63)

Garry Wong, Zi-Qiang Gu, Brian de Costa, Phil Skolnick

Журнал:

European Journal of Pharmacology: Molecular Pharmacology

Рік:

1993

Мова:

english

Файл:

PDF, 638 KB

english, 1993

N-alkyl substituted analogs of the σ receptor ligand BD1008 and traditional σ receptor ligands affect cocaine-induced convulsions and lethality in mice

Rae R. Matsumoto, Kari A. McCracken, Buddy Pouw, Jeffrey Miller, Wayne D. Bowen, Wanda Williams, Brian R. De Costa

Журнал:

Рік:

2001

Мова:

english

Файл:

PDF, 279 KB

english, 2001

Conformationally restricted analogs of BD1008 and an antisense oligodeoxynucleotide targeting σ1 receptors produce anti-cocaine effects in mice

Rae R Matsumoto, Kari A McCracken, Michele J Friedman, Buddy Pouw, Brian R De Costa, Wayne D Bowen

Журнал:

Kari A. McCracken, Wayne D. Bowen, Brian R. de Costa, Rae R. Matsumoto

Рік:

2001

Мова:

english

Файл:

PDF, 574 KB

english, 2001

Two novel σ receptor ligands, BD1047 and LR172, attenuate cocaine-induced toxicity and locomotor activity

Журнал:

François P. Monnet, Brian R. de Costa, Wayne D. Bowen

Рік:

1999

Мова:

english

Файл:

PDF, 418 KB

english, 1999

Differentiation of σ ligand-activated receptor subtypes that modulate NMDA-evoked [3H]-noradrenaline release in rat hippocampal slices

Журнал:

British Journal of Pharmacology

Рік:

1996

Мова:

english

Файл:

PDF, 1.71 MB

english, 1996

Dynorphin A-induced rat hindlimb paralysis and spinal cord injury are not altered by the κ opioid antagonist nor-binaltorphimine

Joseph B. Long, Donald D. Rigamonti, Brian de Costa, Kenner C. Rice, Alberto Martinez-Arizala

Журнал:

Brain Research

Рік:

1989

Мова:

english

Файл:

PDF, 5.80 MB

english, 1989

Neuronal localization of cannabinoid receptors in the basal ganglia of the rat

Miles Herkenham, Allison B. Lynn, Brian R. de Costa, Eric K. Richfield

Журнал:

Brain Research

Рік:

1991

Мова:

english

Файл:

PDF, 4.79 MB

english, 1991

Pharmacological activities of optically pure enantiomers of the κ opioid agonist, U50,488, and its cis diastereomer: evidence for three κ receptor subtypes

Richard B. Rothman, Charles P. France, Victor Bykov, Brian R. De Costa, Arthur E. Jacobson, James H. Woods, Kenner C. Rice

Журнал:

Thomas J. Hudzik, Brian R. De Costa, Donald E. McMillan

Рік:

1989

Мова:

english

Файл:

PDF, 679 KB

english, 1989

σ receptor-mediated emetic response in pigeons: agonists, antagonists and modifiers

Журнал:

Рік:

1993

Мова:

english

Файл:

PDF, 810 KB

english, 1993

Characterization of two novel σ receptor ligands: antidystonic effects in rats suggest σ receptor antagonism

Rae R. Matsumoto, Wayne D. Bowen, Michael A. Tom, Van Nhi Vo, Daniel D. Truong, Brian R. De Costa

Журнал:

Рік:

1995

Мова:

english

Файл:

PDF, 990 KB

english, 1995

Dissociation of the motor effects of (+)-pentazocine from binding to σ1 sites

Rae R. Matsumoto, Wayne D. Bowen, J.Michael Walker, Saundra L. Patrick, Alexander C. Zambon, Van Nhi Vo, Daniel D. Truong, Brian R. De Costa, Kenner C. Rice

Журнал: